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N‑Arylations of Sulfoximines with 2‑Arylpyridines by Copper-Mediated Dual N–H/C–H Activation

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journal contribution
posted on 16.05.2014, 00:00 by Long Wang, Daniel L. Priebbenow, Wanrong Dong, Carsten Bolm
A high-yielding method providing rapid access to new N-arylated sulfoximines has been developed. A stoichiometric amount of copper facilitates the C–H activation of 2-arylpyridines which then undergo oxidative C–N cross-couplings with various sulfoximine derivatives.