Versatile
Synthetic Approach for Selective Diversification of Bicyclic Aza-Diketopiperazines
Version 3 2018-11-19, 17:50
Version 2 2018-11-16, 19:36
Version 1 2018-11-09, 16:33
Posted on 2018-11-19 - 17:50
Herein,
we report a convenient synthesis of unprecedented aza-diketopiperazines
(aza-DKPs). The strategy is based on selective diversification of
bicyclic aza-DKP scaffolds by click reaction, N-acylation, and/or
N-alkylation. These scaffolds containing either azido or amino groups
were obtained by a key Rh(I)-catalyzed hydroformylative cyclohydrocarbonylation
reaction of allyl-substituted aza-DKP. The methodology is readily
amenable to the parallel synthesis of original aza-DKPs to enlarge
the chemical diversity of aza-heterocycles.
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Péron, Florent; Riché, Stéphanie; Lesur, Brigitte; Hibert, Marcel; Breton, Philippe; Fourquez, Jean-Marie; et al. (2018). Versatile
Synthetic Approach for Selective Diversification of Bicyclic Aza-Diketopiperazines. ACS Publications. Collection. https://doi.org/10.1021/acsomega.8b01752
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AUTHORS (8)
FP
Florent Péron
SR
Stéphanie Riché
BL
Brigitte Lesur
MH
Marcel Hibert
PB
Philippe Breton
JF
Jean-Marie Fourquez
NG
Nicolas Girard
DB
Dominique Bonnet