posted on 2006-07-20, 00:00authored byB. V. Subba Reddy, Leleti Rajender Reddy, E. J. Corey
Under special conditions, N-phthaloyl-α-amino acid amides of 8-aminoquinoline can be either acetoxylated or arylated selectively at the β-carbon.
In certain cases, arylation can be effected at the γ-carbon.