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Access to Structurally Diverse Quinoline-Fused Heterocycles via Rhodium(III)-Catalyzed C–C/C–N Coupling of Bifunctional Substrates

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journal contribution
posted on 07.06.2016, 17:21 by Songjie Yu, Yunyun Li, Xukai Zhou, He Wang, Lingheng Kong, Xingwei Li
Rhodium­(III)-catalyzed C–H activation of heteroarenes and functionalization with bifunctional substrates such as anthranils allows facile construction of quinoline-fused heterocycles under redox-neutral conditions. The couplings feature broad substrate scope and provide step-economical access to two classes of quinoline-fused condensed heterocycles.