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A Concise and Convergent Synthesis of PA-824

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journal contribution
posted on 2010-11-05, 00:00 authored by Maurice A. Marsini, Paul J. Reider, Erik J. Sorensen
An efficient four-step synthesis of PA-824, a promising antituberculosis drug candidate, has been developed. This concise approach offers significant improvements over the synthetic route currently used for large-scale production.

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