Access to Structurally Diverse Quinoline-Fused Heterocycles via Rhodium(III)-Catalyzed C–C/C–N Coupling of Bifunctional Substrates
journal contributionposted on 07.06.2016 by Songjie Yu, Yunyun Li, Xukai Zhou, He Wang, Lingheng Kong, Xingwei Li
Any type of content formally published in an academic journal, usually following a peer-review process.
Rhodium(III)-catalyzed C–H activation of heteroarenes and functionalization with bifunctional substrates such as anthranils allows facile construction of quinoline-fused heterocycles under redox-neutral conditions. The couplings feature broad substrate scope and provide step-economical access to two classes of quinoline-fused condensed heterocycles.