ol061389j_si_004.pdf (948.9 kB)
Novel Acetoxylation and C−C Coupling Reactions at Unactivated Positions in α-Amino Acid Derivatives
journal contribution
posted on 2006-07-20, 00:00 authored by B. V. Subba Reddy, Leleti Rajender Reddy, E. J. CoreyUnder special conditions, N-phthaloyl-α-amino acid amides of 8-aminoquinoline can be either acetoxylated or arylated selectively at the β-carbon.
In certain cases, arylation can be effected at the γ-carbon.