jo6b01195_si_002.pdf (3.11 MB)
Iron-Mediated Annulation between Methylene Ketones and Diethanolamines: A Sustainable and Scalable Procedure toward N‑(2-Hydroxyethyl) Pyrroles
journal contribution
posted on 2016-09-07, 00:00 authored by Weiming Hu, Jin-Tao Yu, Dengman Ye, Zhou Zhou, Song Sun, Jiang ChengAn
iron-mediated direct annulation between methylene ketones and diethanolamines
was developed for the efficient synthesis of N-(2-hydroxyethyl)
pyrroles. This protocol shows high efficiency, operational simplicity,
good functional group compatibility as well as broad substrates scope.