Applications of Aziridinium Ions.
Selective Syntheses of
β-Aryl-α,β-diamino Esters

Chuang, Tsung-Hsun; Sharpless, K. Barry

doi:10.1021/ol990256d.s001

ol990256d_si_001.pdf (136.72 kB)

Applications of Aziridinium Ions. Selective Syntheses of β-Aryl-α,β-diamino Esters

journal contribution

posted on 1999-10-06, 00:00 authored by Tsung-Hsun Chuang, K. Barry Sharpless

α,β-Diamino esters are readily prepared through stereospecific and regioselective opening of an aziridinium ion intermediate with a variety of amines. The aziridinium ion is generated from the epoxide in two steps.

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Keywords

esters epoxide Aziridinium aziridinium ion Synthese Ester regioselective variety Ion amines opening stereospecific Aryl Selective Diamino Application

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