@article{Blake2016, author = "James F. Blake and Michael Burkard and Jocelyn Chan and Huifen Chen and Kang-Jye Chou and Dolores Diaz and Danette A. Dudley and John J. Gaudino and Stephen E. Gould and Jonas Grina and Thomas Hunsaker and Lichuan Liu and Matthew Martinson and David Moreno and Lars Mueller and Christine Orr and Patricia Pacheco and Ann Qin and Kevin Rasor and Li Ren and Kirk Robarge and Sheerin Shahidi-Latham and Jeffrey Stults and Francis Sullivan and Weiru Wang and Jianping Yin and Aihe Zhou and Marcia Belvin and Mark Merchant and John Moffat and Jacob B. Schwarz", title = "{Discovery of (S)‑1-(1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl)-4-(2-((1-methyl‑1H‑pyrazol-5-yl)amino)pyrimidin-4-yl)pyridin-2(1H)‑one (GDC-0994), an Extracellular Signal-Regulated Kinase 1/2 (ERK1/2) Inhibitor in Early Clinical Development}", year = "2016", month = "6", url = "https://acs.figshare.com/articles/journal_contribution/Discovery_of_i_S_i_1-_1-_4-Chloro-3-fluorophenyl_-2-hydroxyethyl_-4-_2-_1-methyl_1_i_H_i_pyrazol-5-yl_amino_pyrimidin-4-yl_pyridin-2_1_i_H_i_one_GDC-0994_an_Extracellular_Signal-Regulated_Kinase_1_2_ERK1_2_Inhibitor_in_Early_Clinical_Development/3422317", doi = "10.1021/acs.jmedchem.6b00389.s001" }