One-Pot Sonogashira
Coupling–Cyclization toward Regioselective Synthesis of Benzosultams
Sudarshan Debnath
Shovan Mondal
10.1021/acs.joc.5b00274.s002
https://acs.figshare.com/articles/dataset/One_Pot_Sonogashira_Coupling_Cyclization_toward_Regioselective_Synthesis_of_Benzosultams/2175577
A one-pot
method for the Sonogashira coupling and cyclization of 2-bromobenzenesulfonamides
and terminal alkynes is presented. This method allows access to a
variety of substituted benzosultams regioselectively in excellent
yields. The reasons for regioselectivity are interpreted through density
functional theory (DFT) studies.
2015-04-17 00:00:00
Regioselective Synthesis
terminal alkynes
yield
access
variety
cyclization
BenzosultamsA
method
regioselectivity
DFT
benzosultams regioselectively
density
bromobenzenesulfonamide
Sonogashira